蛋白激酶CK2抑制剂(CX-4945 SODIUM SALT) - Names and Identifiers
蛋白激酶CK2抑制剂(CX-4945 SODIUM SALT) - Physico-chemical Properties
Molecular Formula | C19H13ClN3NaO2
|
Molar Mass | 373.77 |
Solubility | 10 mM in DMSO |
Storage Condition | -20℃ |
蛋白激酶CK2抑制剂(CX-4945 SODIUM SALT) - Preparation solution concentration reference
| 1mg | 5mg | 10mg |
---|
1 mM | 2.69 ml | 13.45 ml | 26.9 ml |
5 mM | 0.538 ml | 2.69 ml | 5.38 ml |
10 mM | 0.269 ml | 1.345 ml | 2.69 ml |
5 mM | 0.054 ml | 0.269 ml | 0.538 ml |
Last Update:2024-01-02 23:10:35
蛋白激酶CK2抑制剂(CX-4945 SODIUM SALT) - Reference Information
biological activity | Silmitasertib sodium salt (CX-4945) is an effective, orally bioavailable, selective inhibitor of casein kinase 2 (CK2), with an IC50 value of 1 nM for CK2α and CK2α. |
target | TargetValue CK2α (cell-free assay) 1 nM CK2α' (cell-free assay) 1 nM |
Target | Value |
CK2α
(Cell-free assay)
| 1 nM |
CK2α'
(Cell-free assay)
| 1 nM |
Last Update:2024-04-10 22:29:15